Synonyms: Celiprolol hydrochloride; (3-[3-Acetyl-4-(3-t-butylamino-2-hydroxypropoxy)phenyl]-2,1-diethylurea hydrochloride; NSC 324509; REV 5320A; ST 1396; Selecor; Tenoloc
Molecular Formula: C20H33N3O4 · HCl
Molecular Weight: 415.95
Linear Structural Formula: C20H33N3O4 · HCl
MDL Number: MFCD00941500
Purity: >=98% (HPLC)
Storage: 2-8C
Biochem Physiol Actions: Celiprolol is a selective adrenoceptor modulator that acts not only as a selective beta1 receptor antagonist, but also as a beta2 receptor partial agonist. Because of its of its beta2 agonist activity, celiprolol lacks the typical side effects of the beta-blockers, such as bronchoconstriction, depression of left ventricular function, and peripheral vasoconstriction, making it a good candidate for patients with both cardiovascular and pulmonary disease. It is currently being investigated for treatment of vascular Ehlers-Danlos Syndrome (vEDS).