Biologically Active Small Molecules, Cayman Chemical, UN2811, 54527-84-3

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54527-84-3 UN2811 Cayman Chemical Biologically Active Small Molecules

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  • Cayman Chemical

    A dihydropyridine L-type calcium channel antagonist that displays antihypertensive and antianginal activity; selectively inhibits adenosine A3 receptors (Ki = 3.25 µM) and CYP3A4 catalytic activity (IC50 = 0.148 µM); activates TRPA1 channels, producing an increase in Ca2+…