Biologically Active Small Molecules, Cayman Chemical, UN2811, 2068-78-2
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Vincristine (sulfate)
Cayman ChemicalAn antimitotic vinca alkaloid which irreversibly blocks mitosis by binding to tubulin (Ki = 85 nM) and inhibiting tubulin polymerization; exported from cells via the ABC transporter P-glycoprotein but not by Mrp1.
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