Biologically Active Small Molecules, Cayman Chemical, 1143573-33-4

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1143573-33-4 Cayman Chemical Biologically Active Small Molecules

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  • Cayman Chemical

    A PPARγ agonist that is 4-fold more potent than rosiglitazone at the PPARγ receptor demonstrating an EC50 value of 0.05 µM; shows high selectivity for PPARγ over PPARα (EC50 = 3.99 µM) or PPARδ (EC50 > 10 µM).