Biologically Active Small Molecules, 132539-06-1

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132539-06-1 Biologically Active Small Molecules

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  • Cayman Chemical

    An antipsychotic, thienobenzodiazepine compound that binds as an antagonist/inverse agonist to dopamine D1 (Ki = 31 nM), dopamine D2 (Ki = 11 nM), dopamine D4 (Ki = 27 nM), serotonin 5-HT2A (Ki = 4 nM), serotonin 5-HT2C (Ki = 11 nM), serotonin 5-HT3 (Ki = 57 nM), muscarinic M1 (Ki = 2 nM),…