LKT Labs, 500 mg
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Citalopram Hydrobromide
LKT LabsCitalopram is a selective serotonin reuptake inhibitor (SSRI) that inhibits the serotonin transporter (SERT); citalopram is clinically used for its antidepressant and anxiolytic activities, although it may prolong the QT interval. The S-isomer of citalopram is active and is sold on its own as…
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Cisplatin
LKT LabsCisplatin is a platinum-based cross-linking agent that exhibits anticancer chemotherapeutic activity. Cisplatin induces crosslinks between guanine bases on DNA; it is clinically used to treat various forms of cancer. In lung cancer cells, cisplatin decreases phosphorylation of PI3K, Akt, and FOXO3a…
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2-tert-Butyl-4-Hydroxyanisole
LKT Labs2-Tert-butyl-4-hydroxyanisole (2-BHA) is one component of butylated hydroxyanisole (BHA). This compound is commonly used as a food additive; it exhibits antioxidative activity. 2-BHA acts as a phase II enzyme inducer, increasing levels of glutathione and glutathione-S-transferase.
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Cilostazol
LKT LabsCilostazol is a quinolone inhibitor of phosphodiesterase 3B (PDE 3B) that exhibits vasodilatory, antiplatelet, anti-inflammatory, anti-diabetic, antidepressant, anxiolytic, and pro-angiogenic activities. Cilostazol is clinically used to treat intermittent claudication associated with peripheral…
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S-(N-Benzylthiocarbamoyl)-L-cysteine
LKT LabsCysteine conjugate of benzyl isothiocyanate, N-dimethylnitrosamine demethylase inhibitor. It induces apoptosis in bladder cancer cells and inhibits cell growth in leukemia cells. Grade: ≥98
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4-tert-Butyl-5-Methoxy-1,2-quinone
LKT Labs4-Tert-butyl-5-methoxy-1,2-quinone exhibits anticancer activity, inhibiting proliferation of leukemia cells.
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This compound is an N-acetyl cysteine conjugate of phenethylisothiocyanate (PEITC-NAC), exhibiting anticancer chemotherapeutic and chemopreventive activities. In lung cancer and prostate cancer models, PEITC-NAC increases activation of JNK, p53, and MAPKs, inducing apoptosis, decreasing tumor…
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Cisatracurium Besylate
LKT LabsCisatracurium is a non-depolarizing neuromuscular junction (NMJ) blocker; it binds the a-d interface of postsynaptic nicotinic acetylcholine receptors (nAChRs). Cisatracurium acts as a skeletal muscle relaxant and is an isomer of parent compound atracurium. Cisatracurium also suppresses atrial…
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3-tert-Butyl-5-Methoxy-1,2-quinone
LKT Labs3-Tert-butyl-5-methoxy-1,2-quinone exhibits anticancer activity, inhibiting proliferation of leukemia cells.