Biologically Active Small Molecules, 101622-51-9, Cayman Chemical

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Cayman Chemical 101622-51-9 Biologically Active Small Molecules

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    An ATP-competitive CDK inhibitor; inhibits CDC2/cyclin B (IC50 = 7 µM), Cdk2/cyclin A (IC50 = 7 µM), Cdk2/cyclin E (IC50 = 7 µM, Cdk/p35 kinase (IC50 = 3 µM), and ERK1/p44 MAPK (IC50 = 25 µM).