Biologically Active Small Molecules, Cayman Chemical, 100 mg, 57808-66-9

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57808-66-9 100 mg Cayman Chemical Biologically Active Small Molecules

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  • Cayman Chemical

    A peripheral dopamine D2 and D3 receptor antagonist (Ki = 0.3 nM; IC50 = 13.6 nM for rat D2 and IC50 = 2.68 nM for rat D3); antiemetic and upper gastrointestinal tract prokinetic activities have been evaluated in clinical trials.