Biologically Active Small Molecules, Cayman Chemical, 183506-66-3
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Apicidin
Cayman ChemicalA fungal toxin that demonstrates selective inhibition of HDAC3/NcoR over HDAC6 (IC50s = 15.8 and 665.1 nM, respectively); has broad spectrum activity against Apicomplexan parasites and exhibits antiproliferative activity against various cancer cell lines (IC50s = 0.13-2.36 μM).
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