A highly potent, selective, non-xanthine adenosine A2A receptor antagonist (Ki = 800 pM for human adenosine A2AR stably expressed in HEK-293 cells).
Synonyms: Adenosine A2A Receptor Antagonist I, ZM 241385 - CAS 139180-30-6 - Calbiochem
Molecular Formula: C16H15N7O2
Molecular Weight: 337.34
Linear Structural Formula: C16H15N7O2
MDL Number: MFCD00908394
Purity: >=98% (HPLC)
Biochem Physiol Actions: Reversible: yes
Legal Information: CALBIOCHEM is a registered trademark of Merck KGaA, Darmstadt, Germany
Other Notes: Poucher, S. M., et al. 1995. Brit. J. Pharmacol. 115, 1096.Ongini, E. et al. 1999. Naunyn Schmiedebergs Arch Pharmacol. 359, 7.Keddie, J. et al. 1996, Eur Journ Pharm. 301, 107.